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Found 3 Enz. Inhib. hit(s) with Target = 'Parathyroid hormone/parathyroid hormone-related peptide receptor' and Ligand = 'BDBM50269979'
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269979(CHEMBL515170 | r-5-(2-E-cyclopropylvinyl)-t-3-ethy...)
Affinity DataIC50:  990nMAssay Description:Displacement of [125I]DPC-AJ1951 from PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269979(CHEMBL515170 | r-5-(2-E-cyclopropylvinyl)-t-3-ethy...)
Affinity DataIC50:  5.78E+3nMAssay Description:Antagonist activity at PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cells assessed as inhibition of DPC-AJ1951-induced cAM...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50269979(CHEMBL515170 | r-5-(2-E-cyclopropylvinyl)-t-3-ethy...)
Affinity DataIC50:  6.80E+4nMAssay Description:Antagonist activity at PTH/PTH-related peptide receptor (unknown origin) expressed in HKRK-B28 cells assessed as inhibition of parathyroid hormone (1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed