Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor gamma' and Ligand = 'BDBM50179244'
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179244(2-{5-[3-methyl-5-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataIC50:  1.37E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179244(2-{5-[3-methyl-5-(7-propyl-3-trifluoromethylbenzo[...)
Affinity DataEC50: >1.00E+4nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed