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Found 1 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM259574'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Amgen

US Patent
LigandPNGBDBM259574(US9505749, 85)
Affinity DataIC50: >8.50E+4nMAssay Description:PARP1 biochemical assay was purchased as a kit from Trevigen (cat.#4676-096-K) and used per manufacturers recommendations.PARP2 biochemical assay was...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent