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Found 2 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50335640'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Cylene Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335640(4-Oxo-4,5-dihydrothieno[3,2-c]quinoline-7-carboxyl...)
Affinity DataIC50:  700nMAssay Description:Inhibition of PARP1 by chemiluminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Cylene Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50335640(4-Oxo-4,5-dihydrothieno[3,2-c]quinoline-7-carboxyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:PARP assays are conducted using a chemiluminescent PARP assay kit (Trevigen). Briefly, reactions are performed in Histone-coated strip wells, by addi...More data for this Ligand-Target Pair
In DepthDetails US Patent