Found 1 Enz. Inhib. hit(s) with Target = 'Poly [ADP-ribose] polymerase 1' and Ligand = 'BDBM50446671'
TargetPoly [ADP-ribose] polymerase 1(Homo sapiens (Human))
Washington University Saint Louis
Curated by ChEMBL
Washington University Saint Louis
Curated by ChEMBL
Affinity DataIC50: 11nMAssay Description:Inhibition of PARP-1 (unknown origin) assessed as NAD+ consumption after 20 mins by fluorometric analysis in presence of activated DNAMore data for this Ligand-Target Pair