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Found 2 Enz. Inhib. hit(s) with Target = 'Prostaglandin D2 receptor' and Ligand = 'BDBM50128699'
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128699((+) (E) 7-[3-(5-Styryl-thiophene-2-sulfonylamino)-...)
Affinity DataIC50:  90nMAssay Description:In vitro inhibition of [3H]- PGD-2 radioligand binding to prostaglandin D2 receptor on human platelet membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor(Homo sapiens (Human))
Shionogi

Curated by ChEMBL
LigandPNGBDBM50128699((+) (E) 7-[3-(5-Styryl-thiophene-2-sulfonylamino)-...)
Affinity DataIC50:  100nMAssay Description:In vitro inhibition of cAMP formation evoked by prostaglandin D2 receptor in human plateletsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed