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Found 4 Enz. Inhib. hit(s) with Target = 'Prostaglandin D2 receptor 2' and Ligand = 'BDBM50309254'
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50309254(2-(4-(4-chlorophenyl)-2-phenylthiazol-5-yl)acetic ...)
Affinity DataIC50:  550nMAssay Description:Displacement of[3H]PGD2 from human CRTH2 receptor expressed in HEK385-7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50309254(2-(4-(4-chlorophenyl)-2-phenylthiazol-5-yl)acetic ...)
Affinity DataIC50:  550nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK285-7 cells assessed as inhibition of beta arrestin translocation by bioluminescence reso...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50309254(2-(4-(4-chlorophenyl)-2-phenylthiazol-5-yl)acetic ...)
Affinity DataIC50:  550nMAssay Description:Displacement of[3H]PGD2 from human CRTH2 receptor expressed in african green monkey COS7 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
7Tm Pharma

Curated by ChEMBL
LigandPNGBDBM50309254(2-(4-(4-chlorophenyl)-2-phenylthiazol-5-yl)acetic ...)
Affinity DataIC50:  960nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in HEK285-7 cells assessed as inhibition of beta arrestin translocation by bioluminescence reso...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed