Affinity DataIC50: 43nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in 293 cells by scintillation counting in presence of 0.5% BSAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.05E+3nMAssay Description:Displacement of [3H]PGD2 from human CRTH2 receptor expressed in 293 cells by scintillation counting in presence of 50% human plasmaMore data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CEM cell assessed as inhibition of PGD2-induced cell migration after 3 hrs by transwell migr...More data for this Ligand-Target Pair