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Found 2 Enz. Inhib. hit(s) with Target = 'Prostaglandin D2 receptor 2' and Ligand = 'BDBM50384473'
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384473(CHEMBL2036222)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3HPGD2 from human CRTH2 receptor expressed in CHO cell membrane after 90 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin D2 receptor 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50384473(CHEMBL2036222)
Affinity DataIC50:  46nMAssay Description:Antagonist activity at human CRTH2 receptor expressed in CHO cell membrane assessed as inhibition of PGD2-induced [35S]GTPgammaS binding after 30 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed