Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with Target = 'Prostate-specific antigen' and Ligand = 'BDBM50434142'
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  72nMpH: 7.8Assay Description:Inhibition of PSA (unknown origin) in 50 mM TRIS.HCL and 100 mM NaCl buffer at pH 7.8More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  72nMAssay Description:Inhibition of human seminal fluid PSA using Mu-SRKSQQY-AMC as substrate measured for 30 mins by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  75nMAssay Description:Inhibition of PSA (unknown origin) in RPMIMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  142nMAssay Description:Inhibition of PSA (unknown origin) in RPMI in presence of 1% fetal bovine serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  604nMAssay Description:Inhibition of PSA (unknown origin) in female plasmaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstate-specific antigen(Homo sapiens (Human))
The Johns Hopkins University

Curated by ChEMBL
LigandPNGBDBM50434142(CHEMBL2381669)
Affinity DataKi:  699nMAssay Description:Inhibition of PSA (unknown origin) in RPMI in presence of 1% fetal bovine serum, 1% penicillin/streptomycin, 1% L-glutamineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed