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Found 2 Enz. Inhib. hit(s) with Target = 'Proteasome subunit beta type-2' and Ligand = 'BDBM50599556'
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50599556(CHEMBL5182479)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of 20S constitutive proteosome beta2c subunit (unknown origin) assessed as substrate hydrolysis using Boc-Leu-Arg-Arg-AMC as fluorogenic s...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50599556(CHEMBL5182479)
Affinity DataKi:  2.00E+4nMAssay Description:Inhibition of 20S immuno proteosome beta2i subunit (unknown origin) assessed as substrate hydrolysis using Boc-Leu-Arg-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
In DepthDetails PubMed