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Found 3 Enz. Inhib. hit(s) with Target = 'Protein AF-9' and Ligand = 'BDBM50459730'
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459730(CHEMBL4211714)
Affinity DataKi:  23nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459730(CHEMBL4211714)
Affinity DataKi:  23nMAssay Description:Binding affinity to MBP-tagged human recombinant AF9 (487 to 568 residues) incubated for 40 mins by measuring fluorescence polarization by microplate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProtein AF-9(Homo sapiens)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459730(CHEMBL4211714)
Affinity DataIC50:  149nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed