Found 1 Enz. Inhib. hit(s) with Target = 'Protein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha' and Ligand = 'BDBM50483440'
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Keio University
Curated by ChEMBL
Keio University
Curated by ChEMBL
Affinity DataIC50: 1.47E+4nMAssay Description:Inhibition of protein farnesyltransferase from human EC17 cells using [3H]FPP and GTP-H-RasMore data for this Ligand-Target Pair