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Found 1 Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha type/glutamine gamma-glutamyltransferase 2' and Ligand = 'BDBM50126829'
TargetProtein kinase C alpha type/glutamine gamma-glutamyltransferase 2(Homo sapiens (Human))
Duke University Medical Center

LigandPNGBDBM50126829((E)-1-(6-(3-acetyl-2,4,6-trihydroxy-5-methylbenzyl...)
Affinity DataIC50:  2.00E+4nMT: 2°CAssay Description:In order to eliminated fluorescence interference, chemicals were subjected to a secondary screening using colorimetric BP incorporation assay. TGase...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed