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Found 5 Enz. Inhib. hit(s) with Target = 'Protein kinase C alpha type' and Ligand = 'BDBM50057509'
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  15nMAssay Description:Displacement of phorbol 12,13-dibutyrate (PDBU) from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  15nMAssay Description:Displacement phorbol 12,13-dibutyrate(PDBU) binding from recombinant Protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  15nMAssay Description:Displacement of PDBU from recombinant Protein kinase C alpha with phosphatidylserineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  15nMAssay Description:Displacement of [3H]- PDBu from recombinant PKC alpha expressed in baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Institute Of Organic Chemistry

Curated by ChEMBL
LigandPNGBDBM50057509((2S,5S)-8-Dec-1-ynyl-5-hydroxymethyl-2-isopropyl-1...)
Affinity DataKi:  23nMAssay Description:Inhibition of [3H]-phorbol 12,13-dibutyrate (PDBu) binding to human recombinant protein kinase C alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed