Found 1 Enz. Inhib. hit(s) with Target = 'Protein mono-ADP-ribosyltransferase PARP4' and Ligand = 'BDBM50503853'
TargetProtein mono-ADP-ribosyltransferase PARP4(Homo sapiens (Human))
Oregon Health And Science University
Curated by ChEMBL
Oregon Health And Science University
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human PARP4 BRCT-catalytic domain (1 to 572 residues) assessed as reduction in MARylation of SRPK2 substrate after 60 mins in presence ...More data for this Ligand-Target Pair