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Found 2 Enz. Inhib. hit(s) with Target = 'RAC-alpha serine/threonine-protein kinase' and Ligand = 'BDBM11823'
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM11823(Azepane Derivative 4 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  4nMAssay Description:Inhibition of PKBalpha (unknown origin) expressed in Sf9 insect cells using Biotin-SGRARTSSFAEPG as substrate after 30 mins by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRAC-alpha serine/threonine-protein kinase(Homo sapiens (Human))
Wuhan Institute Of Technology

Curated by ChEMBL
LigandPNGBDBM11823(Azepane Derivative 4 | N-((3R,4R)-4-{[4-(2-fluoro-...)
Affinity DataIC50:  4nMpH: 7.5 T: 2°CAssay Description:An ELISA-based assay has been developed for the serine/threonine kinase, PKB-alpha. The assay utilizes an N-terminally biotinylated substrate peptide...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed