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Found 1 Enz. Inhib. hit(s) with Target = 'RAC-beta serine/threonine-protein kinase' and Ligand = 'BDBM24878'
TargetRAC-beta serine/threonine-protein kinase(Homo sapiens (Human))
Merck Research Laboratories

LigandPNGBDBM24878(6-phenyl-7-[4-({4-[5-(pyridin-2-yl)-4H-1,2,4-triaz...)
Affinity DataIC50:  59nMAssay Description:Purified recombinant human Akt kinase was monitored for kinase activity in the presence or absence of inhibitors in a 96-well format. Detection was d...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed