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Found 1 Enz. Inhib. hit(s) with Target = 'RAC-gamma serine/threonine-protein kinase' and Ligand = 'BDBM50427337'
TargetRAC-gamma serine/threonine-protein kinase(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50427337(CHEMBL2325991)
Affinity DataIC50:  2.89E+3nMAssay Description:Inhibition of recombinant Akt3 (unknown origin) using 5-FAM-labeled peptide as substrate after 1 hr by caliper off-chip incubation mobility shift ass...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed