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Found 3 Enz. Inhib. hit(s) with Target = 'Relaxin-3 receptor 1' and Ligand = 'BDBM50534453'
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534453(CHEMBL4557279)
Affinity DataKi:  275nMAssay Description:Displacement of Eu-H3/15 from human RXFP3 receptor expressed in CHOK1 cells by time-resolved fluorescent whole cell binding assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534453(CHEMBL4557279)
Affinity DataEC50:  3.30nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells cotransfected with beta-galactosidase assessed as inhibition of forskolin-stimulate...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetRelaxin-3 receptor 1(Homo sapiens (Human))
Kobe Gakuin University

Curated by ChEMBL
LigandPNGBDBM50534453(CHEMBL4557279)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at human RXFP3 receptor expressed in CHOK1 cells assessed as ERK1/2 phosphorylation incubated for 5 mins by alphascreen surefire ass...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed