Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor RXR-gamma' and Ligand = 'BDBM50122348'
TargetRetinoic acid receptor RXR-gamma(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50122348((2E,4E)-6-[1-(3,5-Di-tert-butyl-phenyl)-cyclopropy...)
Affinity DataKd:  16nMAssay Description:Inhibition of [3H]-9-cis-RA binding to human Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRetinoic acid receptor RXR-gamma(Mus musculus)
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50122348((2E,4E)-6-[1-(3,5-Di-tert-butyl-phenyl)-cyclopropy...)
Affinity DataEC50:  23nMAssay Description:Transcriptional activation in CV-1 cells expresing mouse Retinoid X receptor RXR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed