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Found 3 Enz. Inhib. hit(s) with Target = 'Reverse transcriptase/RNaseH' and Ligand = 'BDBM50050637'
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050637((8-Ethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azulen...)
Affinity DataIC50:  2.19E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rN.dN template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050637((8-Ethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azulen...)
Affinity DataIC50:  3.90E+3nMAssay Description:Ability to inhibit HIV-1 IIIB reverse transcriptase catalyzed incorporation of tritiated thymidine triphosphate onto a biotinylated rA.dT template pr...More data for this Ligand-Target Pair
In DepthDetails Article
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
TBA

Curated by ChEMBL
LigandPNGBDBM50050637((8-Ethyl-8H-1,3a,7,8,9-pentaaza-dibenzo[e,h]azulen...)
Affinity DataIC50:  3.90E+3nMAssay Description:Inhibitory activity against HIV-1 reverse transcriptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed