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Found 3 Enz. Inhib. hit(s) with Target = 'Ribosomal protein S6 kinase alpha-5' and Ligand = 'BDBM50601147'
TargetRibosomal protein S6 kinase alpha-5(Homo sapiens (Human))
Ucb

Curated by ChEMBL
LigandPNGBDBM50601147(CHEMBL5183977)
Affinity DataIC50:  79nMAssay Description:Inhibition of full-length N-terminal His-TEV-tagged inactive form of MSK1 (2 to 802 residues) (unknown origin) expressed in HEK293 cells using FAM-PS...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRibosomal protein S6 kinase alpha-5(Homo sapiens (Human))
Ucb

Curated by ChEMBL
LigandPNGBDBM50601147(CHEMBL5183977)
Affinity DataIC50:  794nMAssay Description:Inhibition of N-terminal His-Smt-tagged MSK1 C-terminal kinase domain (414 to 738 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetRibosomal protein S6 kinase alpha-5(Homo sapiens (Human))
Ucb

Curated by ChEMBL
LigandPNGBDBM50601147(CHEMBL5183977)
Affinity DataIC50:  794nMAssay Description:Inhibition of N-terminal His-Smt-tagged MSK1 C-terminal kinase domain (414 to 738 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3)...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed