Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase TAO2' and Ligand = 'BDBM2579'
TargetSerine/threonine-protein kinase TAO2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 3.5nMAssay Description:Inhibition of human TAOK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataIC50: 11.7nMAssay Description:Inhibition of human TAOK2 using MBP as substrate by [gamma-33P]-ATP assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein kinase TAO2(Homo sapiens (Human))
Beijing Normal University
Curated by ChEMBL
Beijing Normal University
Curated by ChEMBL
Affinity DataKd: 12nMAssay Description:Binding constant for TAOK2 kinase domainMore data for this Ligand-Target Pair