Affinity DataKi: 6nMAssay Description:Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 receptor binding site by using [3H]- DOB as a radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 7.80nMAssay Description:Binding affinity for the Opioid receptor kappa 1More data for this Ligand-Target Pair
Affinity DataKi: 560nMAssay Description:Binding affinity to rat cortical membranes at 5-hydroxytryptamine 2 (5-HT2) receptor using [3H]KET as a radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 930nMAssay Description:Effect on plasma amine oxidase (0.1 uM) after 15 min of incubation at pH 7.2More data for this Ligand-Target Pair
Affinity DataKi: 950nMAssay Description:Binding affinity was determined against 5-hydroxytryptamine 2 receptor from male Sprague-Dawley rat brain.More data for this Ligand-Target Pair
Affinity DataKi: 977nMAssay Description:Displacement of [3H]ketanserin from 5-hydroxytryptamine 2 receptor of rat frontal cortex homogenateMore data for this Ligand-Target Pair
Affinity DataKi: 2.95E+3nMAssay Description:Binding affinity to 5-hydroxytryptamine 2 receptor in rat frontal cortical membranes by [3H]- KET displacement.More data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Binding affinity of the compound against 5-hydroxytryptamine 1A receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 3.60E+3nMAssay Description:Binding affinity against 5-hydroxytryptamine 2 receptor using [3H]ket as radioligand.More data for this Ligand-Target Pair
Affinity DataIC50: 4.60E+3nMAssay Description:Compound was evaluated for its inhibitory activity against 5-hydroxytryptamine 2 receptor of rat anterior cortex using [3H]ketanserin as the radiolig...More data for this Ligand-Target Pair
TargetSerotonin 2 (5-HT2) receptor(Homo sapiens (Human))
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Smithkline Beecham Pharmaceuticals
Curated by ChEMBL
Affinity DataKd: 3.16E+3nMAssay Description:Binding affinity for 5-hydroxytryptamine 2 receptor was determinedMore data for this Ligand-Target Pair