Affinity DataKi: 7.90nMAssay Description:Binding affinity at 5-hydroxytryptamine 2 receptor from striata wistar rats by [3H]ketanserin displacement.More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of 5-hydroxytryptamine 2 induced vasoconstriction of rat caudal artery.More data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Antagonistic activity against 5-hydroxytryptamine 2 receptor on rat frontal cortex membrane.More data for this Ligand-Target Pair