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Found 3 Enz. Inhib. hit(s) with Target = 'Sigma non-opioid intracellular receptor 1' and Ligand = 'BDBM50044725'
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Esteve

Curated by ChEMBL
LigandPNGBDBM50044725(1-[2-(3,4-Dichloro-phenyl)-ethyl]-4-methyl-piperaz...)
Affinity DataKi:  6.30nMAssay Description:Displacement of [3H](+)pentazocine from human sigma 1 receptor transfected in HEK293 cell membranes after 120 mins by scintillation counterMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
Esteve

Curated by ChEMBL
LigandPNGBDBM50044725(1-[2-(3,4-Dichloro-phenyl)-ethyl]-4-methyl-piperaz...)
Affinity DataKi:  9.20nMAssay Description:Ability to displace [3H](+)-pentazocine at sigma receptor in guinea pig brain membrane was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSigma non-opioid intracellular receptor 1(Cavia porcellus (Guinea pig))
Universit£

Curated by ChEMBL
LigandPNGBDBM50044725(1-[2-(3,4-Dichloro-phenyl)-ethyl]-4-methyl-piperaz...)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-(+)-pentazocine from Dunkin-Hartley guinea pig brain cortex Sigma 1 receptor incubated for 150 mins by liquid scintillation coun...More data for this Ligand-Target Pair
In DepthDetails PubMed