Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50046736'
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Yale School Of Medicine
Curated by ChEMBL
Yale School Of Medicine
Curated by ChEMBL
Affinity DataKi: 100nMAssay Description:Binding affinity to dopamine transporter (DAT) in rat forebrain tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Yale School Of Medicine
Curated by ChEMBL
Yale School Of Medicine
Curated by ChEMBL
Affinity DataKi: 182nMAssay Description:Binding affinity to dopamine transporter in membranes of cells selectively expressing the human genes for DATMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Yale School Of Medicine
Curated by ChEMBL
Yale School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:In vitro inhibitory activity against radioligand [3H]-WN 35,428 binding to dopamine transporter (DAT) in rat striatal tissueMore data for this Ligand-Target Pair
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Yale School Of Medicine
Curated by ChEMBL
Yale School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of [3H]3-beta-(4-fluorophenyl)tropane-2beta-carboxylic acid methyl ester binding to dopamine transporter of cynomolgus monkey striatumMore data for this Ligand-Target Pair