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Found 4 Enz. Inhib. hit(s) with Target = 'Sodium-dependent dopamine transporter' and Ligand = 'BDBM50136674'
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50136674((3R)-N-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propa...)
Affinity DataKi:  550nMAssay Description:Displacement of [125I]RTI-55 from human recombinant DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50136674((3R)-N-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propa...)
Affinity DataKi:  659nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Eli Lilly

Curated by PDSP Ki Database
LigandPNGBDBM50136674((3R)-N-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propa...)
Affinity DataIC50:  660nMAssay Description:Displacement of [125I]RTI55 from DAT in Sprague-dawley rat striatum by liquid scintillation spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Human Biomolecular Research Institute

Curated by ChEMBL
LigandPNGBDBM50136674((3R)-N-methyl-3-(1-naphthyloxy)-3-(2-thienyl)propa...)
Affinity DataIC50:  809nMAssay Description:Inhibition of [3H]DA reuptake at human DAT expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed