Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Sodium-dependent serotonin transporter' and Ligand = 'BDBM50135246'
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50135246((S)-1-((2S,4R)-4-(benzo[b]thiophen-2-yl)-2-methylp...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity at 5-HT reuptake site labeled with [3H]-paroxetineMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50135246((S)-1-((2S,4R)-4-(benzo[b]thiophen-2-yl)-2-methylp...)
Affinity DataKi:  0.530nMAssay Description:Displacement of [3H]paroxetine from 5HT reuptake siteMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Eli Lilly

Curated by ChEMBL
LigandPNGBDBM50135246((S)-1-((2S,4R)-4-(benzo[b]thiophen-2-yl)-2-methylp...)
Affinity DataKi:  0.530nMAssay Description:Affinity at the 5-HT reuptake site labeled with [3H]-paroxetine using rat frontal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed