Found 2 Enz. Inhib. hit(s) with Target = 'Solute carrier organic anion transporter family member 1B1' and Ligand = 'BDBM50391000'
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Hospital
Curated by ChEMBL
University Hospital
Curated by ChEMBL
Affinity DataKi: 2.00E+3nMAssay Description:TP_TRANSPORTER: inhibition of BSP uptake in Xenopus laevis oocytesMore data for this Ligand-Target Pair
TargetSolute carrier organic anion transporter family member 1B1(Homo sapiens (Human))
University Hospital
Curated by ChEMBL
University Hospital
Curated by ChEMBL
Affinity DataIC50: 230nMAssay Description:TP_TRANSPORTER: inhibition of estradiol-17beta-glucuronide uptake(estradiol-17beta-glucuronide:0.02uM) in OATP1B1-expressing HEK293 cellsMore data for this Ligand-Target Pair