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Found 1 Enz. Inhib. hit(s) with Target = 'Solute carrier organic anion transporter family member 1B3' and Ligand = 'BDBM50339127'
TargetSolute carrier organic anion transporter family member 1B3(Homo sapiens (Human))
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50339127((3S,6S,9S,12R,15S,18S,21S,24S,27R,30S,33S)-25,30-d...)
Affinity DataIC50:  220nMAssay Description:Inhibition of OATP1B3 (unknown origin) expressed in HEK293 cells using [3H]estradiol-17beta-glucuronide substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed