Compile Data Set for Download or QSAR
maximum 50k data
Found 10 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 3' and Ligand = 'BDBM50389590'
TargetSomatostatin receptor type 3(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  8.90nMAssay Description:Displacement of [125I]SS-14 from mouse SST3 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  8.90nMAssay Description:Displacement of [125I]SS-28 from mouse SSTR3 transfected in CHO cells after 60 to 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  11nMAssay Description:Inhibition of human SSTR3 transfected in CHO cells assessed as inhibition of SRIF-induced reduction of cAMP accumulation after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]SS-14 from human SST3 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  14nMAssay Description:Binding affinity to human somatostatin receptor type 3More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  14nMAssay Description:Displacement of [125I]SS-28 from human SSTR3 transfected in CHO cells after 60 to 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  16nMAssay Description:Inhibition of mouse SSTR3 transfected in CHO cells assessed as inhibition of SRIF-induced reduction of cAMP accumulation after 45 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(MOUSE)
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  16nMAssay Description:Antagonist activity at mouse SST3 receptor expressed in CHO cells assessed as inhibition of forskolin/SS-14-stimulated cAMP accumulation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataIC50:  22nMAssay Description:Antagonist activity at human SST3 receptor expressed in CHO cells assessed as inhibition of forskolin/SS-14-stimulated cAMP accumulation preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 3(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50389590(CHEMBL2069502)
Affinity DataEC50:  22nMAssay Description:Antagonist activity at human somatostatin receptor type 3 assessed as inhibition of cAMP levelsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed