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Found 3 Enz. Inhib. hit(s) with Target = 'Somatostatin receptor type 5' and Ligand = 'BDBM50227111'
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227111(CHEMBL236587 | N-(1-(3-ethoxy-4-methoxybenzyl)pipe...)
Affinity DataKi:  121nMAssay Description:Displacement of [125I]11-Tyr somatostatin-14 from human SST5R expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227111(CHEMBL236587 | N-(1-(3-ethoxy-4-methoxybenzyl)pipe...)
Affinity DataKi:  121nMAssay Description:Displacement of SST14 from human recombinant SST5 receptor expressed in CHO cells by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 5(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50227111(CHEMBL236587 | N-(1-(3-ethoxy-4-methoxybenzyl)pipe...)
Affinity DataIC50:  740nMAssay Description:Antagonist activity at human SST5R expressed in CHO cells assessed as reversal of somatostatin-14 induced cAMP responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed