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Found 2 Enz. Inhib. hit(s) with Target = 'Stearoyl-CoA desaturase' and Ligand = 'BDBM50304955'
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50304955(CHEMBL590108 | N-(2-hydroxy-2-(thiophen-3-yl)ethyl...)
Affinity DataIC50:  7nMAssay Description:Inhibition of Scd1 in human HEK-293A cell microsomes assessed as conversion of [14C]stearate to [14C]oleate pretreated for 10 mins measured after 60 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetStearoyl-CoA desaturase(Homo sapiens (Human))
Daiichi Sankyo

Curated by ChEMBL
LigandPNGBDBM50304955(CHEMBL590108 | N-(2-hydroxy-2-(thiophen-3-yl)ethyl...)
Affinity DataIC50:  21nMAssay Description:Inhibition of human Scd1 expressed in HEK-293A cells assessed as conversion of [14C]stearate to [14C]oleate pretreated for 30 mins measured after 4 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed