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Found 3 Enz. Inhib. hit(s) with Target = 'Synaptic vesicular amine transporter' and Ligand = 'BDBM50359499'
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50359499((S)Methamphetamine | METHAMPHETAMINE)
Affinity DataKi:  2.46E+3nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat brain synaptic vesicles by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50359499((S)Methamphetamine | METHAMPHETAMINE)
Affinity DataKi:  2.46E+3nMAssay Description:Inhibition of VMAT2-mediated [3H]-dopamine uptake in rat striata isolated synaptic vesicles by liquid scintillation spectroscopyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Kentucky

Curated by ChEMBL
LigandPNGBDBM50359499((S)Methamphetamine | METHAMPHETAMINE)
Affinity DataKi:  8.01E+4nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in rat whole brain by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed