Affinity DataIC50: 27nMAssay Description:Antagonist activity at mouse prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
Affinity DataIC50: 61nMAssay Description:Antagonist activity at human prostanoid TP receptor expressed in QBI-HEK 293A cells assessed as inhibition of 1-BOP-induced increase in inositol mono...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of human TP receptor expressed in QBI-HEK 293A cells assessed as IP3 metabolite level after 1 hr by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 523nMAssay Description:Antagonist activity against human thromboxane A2 receptor alpha expressed in QBI-HEK293A cells assessed as reduction in I-BOP-induced inositol monoph...More data for this Ligand-Target Pair
Affinity DataKd: 141nMAssay Description:Displacement of [3H]SQ-29548 from human prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair
Affinity DataKd: 26nMAssay Description:Displacement of [3H]SQ-29548 from mouse prostanoid TP receptor expressed in QBI-HEK 293A cells after 2 hrs by scintillation proximity assayMore data for this Ligand-Target Pair