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Found 3 Enz. Inhib. hit(s) with Target = 'Thyroid hormone receptor alpha' and Ligand = 'BDBM50178970'
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50178970(6-(4-hydroxy-3-isopropylphenoxy)-5,7-dimethylquino...)
Affinity DataIC50:  200nMAssay Description:Inhibition of human TRalpha1 by radioligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50178970(6-(4-hydroxy-3-isopropylphenoxy)-5,7-dimethylquino...)
Affinity DataIC50:  200nMAssay Description:Inhibition of thyroid hormone receptor alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
Karo Bio

Curated by ChEMBL
LigandPNGBDBM50178970(6-(4-hydroxy-3-isopropylphenoxy)-5,7-dimethylquino...)
Affinity DataEC50:  83nMAssay Description:Efficacy against TRAF-alpha-1 reporter cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed