Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Toll-like receptor 2' and Ligand = 'BDBM50399455'
TargetToll-like receptor 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50399455(CHEMBL2179402)
Affinity DataKi:  25nMAssay Description:Displacement of Eu-DTPA from human TLR2 expressed in SU.86.86 cells after 1 hrMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 2(Homo sapiens (Human))
H. Lee Moffitt Cancer Center And Research Institute

Curated by ChEMBL
LigandPNGBDBM50399455(CHEMBL2179402)
Affinity DataEC50:  39nMAssay Description:Agonist activity at human TLR2 expressed in HEK293 cells assessed as induction of NF-kappaB signaling after 24 hrs by luminescence based luciferase r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed