Found 2 Enz. Inhib. hit(s) with Target = 'Trace amine-associated receptor 1' and Ligand = 'BDBM122294'
Affinity DataKi: 1.70nM ΔG°: -46.5kJ/moleT: 2°CAssay Description:Binding assay was performed at 4 C. in a final volume of 1 ml, and with an incubation time of 30 min. The radioligand [3H]-rac-2-(1,2,3,4-tetrahydro-...More data for this Ligand-Target Pair
TargetTrace amine-associated receptor 1(Homo sapiens (Human))
Roche Innovation Center Basel
Curated by ChEMBL
Roche Innovation Center Basel
Curated by ChEMBL
Affinity DataEC50: 9nMAssay Description:Agonist activity at human TAAR1 expressed in recombinant HEK293 cells assessed as cAMP accumulation after 30 mins by luminometerMore data for this Ligand-Target Pair