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Found 1 Enz. Inhib. hit(s) with Target = 'Transcription factor Jun' and Ligand = 'BDBM50092872'
TargetTranscription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50092872(2-Chloro-4-ethyl-pyrimidine-5-carboxylic acid (3,5...)
Affinity DataIC50:  300nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed