Compile Data Set for Download or QSAR
maximum 50k data
Found 1 Enz. Inhib. hit(s) with Target = 'Transcription factor Jun' and Ligand = 'BDBM50092890'
TargetTranscription factor Jun(Homo sapiens (Human))
Signal Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50092890(2-Chloro-pyrimidine-5-carboxylic acid (3,5-bis-tri...)
Affinity DataIC50:  300nMAssay Description:Concentration required to inhibit activator protein-1(AP-1) mediated transcriptional activation in human Jurkat T-cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed