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Found 1 Enz. Inhib. hit(s) with Target = 'Transforming growth factor beta-1 proprotein' and Ligand = 'BDBM50184872'
TargetTransforming growth factor beta-1 proprotein(Homo sapiens (Human))
Monash University

Curated by ChEMBL
LigandPNGBDBM50184872(4-(4-(3-(pyridin-2-yl)-1H-pyrazol-4-yl)pyridin-2-y...)
Affinity DataIC50:  446nMAssay Description:Inhibition of TGF-beta1 signaling in human HEK293 cells transfected with luciferase and FAST-2 gene expression vector A3-LUX after 16 hrs by lucifera...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed