Found 4 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily A member 1' and Ligand = 'BDBM50061117'
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 210nMAssay Description:Agonist activity at TRPA1 (unknown origin) channel desensitization in presence of icilinMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Agonist activity at TRPA1 (unknown origin) channel desensitization in presence of isothiocyanateMore data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Rattus norvegicus)
University Of Eastern Piedmont
Curated by ChEMBL
University Of Eastern Piedmont
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Agonist activity at recombinant rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo4-AM probe based fluor...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Homo sapiens (Human))
Scientus Pharma
Curated by ChEMBL
Scientus Pharma
Curated by ChEMBL
Affinity DataEC50: 180nMAssay Description:Agonist activity at TRPA1 (unknown origin) activationMore data for this Ligand-Target Pair