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Found 4 Enz. Inhib. hit(s) with Target = 'Transient receptor potential cation channel subfamily V member 1' and Ligand = 'BDBM50169728'
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50169728(CHEMBL364193 | N-(4-tert-Butyl-benzyl)-2-(3-fluoro...)
Affinity DataKi:  118nMAssay Description:Antagonist activity towards rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50169728(CHEMBL364193 | N-(4-tert-Butyl-benzyl)-2-(3-fluoro...)
Affinity DataKi:  118nMAssay Description:Antagonist activity at rat TRPV1 receptor expressed in CHO cells assessed as decrease in capsaicin-induced intracellular 45Ca2+ uptake after 1 hr by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50169728(CHEMBL364193 | N-(4-tert-Butyl-benzyl)-2-(3-fluoro...)
Affinity DataKi:  470nMAssay Description:Displacement of [3H]RTX from rat TRPV1 receptor expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 1(Rattus norvegicus (rat))
Seoul National University

Curated by ChEMBL
LigandPNGBDBM50169728(CHEMBL364193 | N-(4-tert-Butyl-benzyl)-2-(3-fluoro...)
Affinity DataKi:  472nMAssay Description:In vitro inhibition of [3H]-RTX binding to rat TRPV1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed