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Found 2 Enz. Inhib. hit(s) with Target = 'Tryptase beta-2/delta/gamma' and Ligand = 'BDBM50093187'
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Axys Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50093187(1,5-di{4-[4-amino(imino)methylbenzylcarbamoyl]hexa...)
Affinity DataKi:  8.70nMAssay Description:Binding affinity to 5-HT3 serotonin receptor in NG 108-15 neuroblastoma glioma cells using [3H]-GR-65,630 radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
Axys Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50093187(1,5-di{4-[4-amino(imino)methylbenzylcarbamoyl]hexa...)
Affinity DataKi:  9nMAssay Description:Evaluated for its inhibitory potency against tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed