Found 8 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50042235'
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Binding affinity to AT1 receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Inhibitory concentration against angiotensin II receptor, type 1More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Compound was evaluated for its binding affinity towards human Angiotensin II receptor, type 1More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Binding affinity against AT1 in human hepatoma cell line, PLC-PRF-5More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:In vitro binding affinity towards Angiotensin II receptor, type 1 of human hepatoma cell line PLC-PRF-5More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 0.900nMAssay Description:Displacement of [125I]- Ang II from type 1 Angiotensin II receptorMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 6nMAssay Description:Antagonist activity at human AT1 overexpressed in CHO-K1 cells in presence of 10 nM [Val5-angiotensin II measured after 90 mins by HTRF based IP-one ...More data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
National Heart And Lung Institute
Curated by ChEMBL
National Heart And Lung Institute
Curated by ChEMBL
Affinity DataIC50: 20.8nMAssay Description:Binding affinity to angiotensin AT1 receptorMore data for this Ligand-Target Pair