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Found 4 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50049186'
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (Bau)

Curated by ChEMBL
LigandPNGBDBM50049186((S)-3-Methyl-2-{pentanoyl-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I-Sar1-Ile8]-Ang2 from human angiotensin 2 receptor type 1 receptor expressed in HEK293 cells after 1 hr by gamma counting analys...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (Bau)

Curated by ChEMBL
LigandPNGBDBM50049186((S)-3-Methyl-2-{pentanoyl-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition constant against Angiotensin II receptor, type 1 was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (Bau)

Curated by ChEMBL
LigandPNGBDBM50049186((S)-3-Methyl-2-{pentanoyl-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataIC50:  2.70nMAssay Description:Tested for inhibition of Angiotensin II receptor, type 1 in the absence of bovine serum albumin (BSA)More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Bahcesehir University (Bau)

Curated by ChEMBL
LigandPNGBDBM50049186((S)-3-Methyl-2-{pentanoyl-[2'-(1H-tetrazol-5-yl)-b...)
Affinity DataIC50:  7.40nMAssay Description:Displacement of [125-I]-[Sar1, AngII from AT1R (unknown origin) expressed in Escherichia coli BL 21 (DE3) incubated for 2 hrs by radioimmunoassayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed