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Found 3 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50049200'
TargetType-1 angiotensin II receptor(Bos taurus)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049200(2-Ethyl-5,7-dimethyl-3-[9-(1H-tetrazol-5-ylmethyl)...)
Affinity DataIC50:  11nMAssay Description:Binding affinity to angiotensin AT1 receptor in bovine adrenal cortex membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(Bos taurus)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049200(2-Ethyl-5,7-dimethyl-3-[9-(1H-tetrazol-5-ylmethyl)...)
Affinity DataIC50:  11nMAssay Description:In vitro antagonistic potency against Angiotensin II receptor, type 1 in rat adrenal cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
The M. S. University Of Baroda

Curated by ChEMBL
LigandPNGBDBM50049200(2-Ethyl-5,7-dimethyl-3-[9-(1H-tetrazol-5-ylmethyl)...)
Affinity DataKd:  0.631nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortic strip assessed as inhibition of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed