Found 3 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM50049200'
Affinity DataIC50: 11nMAssay Description:Binding affinity to angiotensin AT1 receptor in bovine adrenal cortex membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:In vitro antagonistic potency against Angiotensin II receptor, type 1 in rat adrenal cortexMore data for this Ligand-Target Pair
Affinity DataKd: 0.631nMAssay Description:Antagonist activity at angiotensin AT1 receptor in rabbit aortic strip assessed as inhibition of angiotensin 2-induced contractile responseMore data for this Ligand-Target Pair