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Found 10 Enz. Inhib. hit(s) with Target = 'Type-1 angiotensin II receptor' and Ligand = 'BDBM82433'
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1nMAssay Description:In vitro binding affinity determined by its ability to displace the specific binding ligand [125I]-Sar1, Ile8-AII from Angiotensin II receptor, type ...More data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.5nMAssay Description:In vivo inhibitory concentration of the compound against Angiotensin II receptor, type 1 of rabbit aorta membraneMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.5nMAssay Description:Inhibition of [125I]-Sar1-Ile8-Ang II binding to Angiotensin II receptor type 1 from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.70nMAssay Description:Inhibitory concentration against angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of Angiotensin II receptor, type 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.70nMAssay Description:Tested for in vitro binding affinity against angiotensin I (AT1) receptor to competitively block the specific binding of [125I]- [Sar1,Ile8] AII to a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.70nMAssay Description:In vitro inhibitory activity against Angiotensin II receptor, type 1 in rabbit aorta membrane preparations.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.70nMAssay Description:Binding affinity against AT-1 receptor from rabbit aorta using [125I]-Sar1-Ile8-Ang II without BSAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetType-1 angiotensin II receptor(RABBIT)
TBA

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  1.70nMAssay Description:In vitro ability of the compound to inhibit the binding of radioligand 125I[Sar1,IIe8]AII to AT1 receptor from rabbit aortaMore data for this Ligand-Target Pair
In DepthDetails Article
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
Organon Laboratories

Curated by ChEMBL
LigandPNGBDBM82433(CHEMBL302102 | L-159,689 | L-159689 | N-Pentyl-N-[...)
Affinity DataIC50:  7nMAssay Description:In vivo inhibitory concentration of the compound against Angiotensin II receptor, type 1 of rat adrenal membraneMore data for this Ligand-Target Pair
In DepthDetails Article